Benzazoles: I. Regioselective arylsulfonylation of benzimidazol-2-amine View Full Text


Ontology type: schema:ScholarlyArticle     


Article Info

DATE

2013-01

AUTHORS

T. N. Kaipnazarov, K. B. Abdireimov, N. S. Mukhamedov, R. Ya. Okmanov, B. Tashkhodjaev, G. E. Berdimbetova, Kh. M. Shakhidoyatov

ABSTRACT

Benzimidazol-2-amine reacted with arenesulfonyl chlorides in the presence of triethylamine in regioselective fashion at the endocyclic nitrogen atom, the exocyclic amino group remaining intact. The yields of 1-arylsulfonylbenzimidazol-2-amines depend on the electronic properties of substituents in the benzene ring of arenesulfonyl chlorides.

PAGES

108-111

References to SciGraph publications

  • 2006-05. Synthesis and tuberculostatic activity of new benzimidazole derivatives in CHEMISTRY OF HETEROCYCLIC COMPOUNDS
  • Identifiers

    URI

    http://scigraph.springernature.com/pub.10.1134/s1070428013010181

    DOI

    http://dx.doi.org/10.1134/s1070428013010181

    DIMENSIONS

    https://app.dimensions.ai/details/publication/pub.1030820252


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