Synthesis of sodium 5-sulfate-ivermectin and disodium 4″,5-disulfate-ivermectin View Full Text


Ontology type: schema:ScholarlyArticle     


Article Info

DATE

2018-05

AUTHORS

M. A. Shchetinina, E. I. Chernoburova, N. G. Kolotyrkina, M. Kh. Dzhafarov, F. I. Vasilevich, I. V. Zavarzin

ABSTRACT

Treatment of ivermectin with sulfuric acid–acetic anhydride in pyridine gives sodium 5-sulfate-ivermectin and disodium 4″,5-disulfate-ivermectin. The synthesized salts are water-soluble compounds with promising antiparasitic activity.

PAGES

836-839

Identifiers

URI

http://scigraph.springernature.com/pub.10.1007/s11172-018-2146-z

DOI

http://dx.doi.org/10.1007/s11172-018-2146-z

DIMENSIONS

https://app.dimensions.ai/details/publication/pub.1106255451


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