Synthesis of polyazaheterocycles containing linearly bound 1,2,4-thiadiazole using enaminones View Full Text


Ontology type: schema:ScholarlyArticle     


Article Info

DATE

2016-04

AUTHORS

Kh. S. Shikhaliev, P. S. Romanov, A. S. Shestakov, N. V. Stolpovskaya, M. Yu. Krysin, A. Yu. Potapov, A. N. Proshin

ABSTRACT

A reaction of N-substituted 5-amino-3-(2-oxopropyl)-1,2,4-thiadiazoles with dimethylformamide dimethyl acetal gave 3-(5-amino-1,2,4-thiadiazol-3-yl)-4-(dimethylamino)but-3en-2-ones, whose cyclization with hydrazine, guanidine, 1H-pyrazol-5-amines and 6-aminopyrimidin-4(3H)-ones led to 3-methyl-1H-pyrazole, 4-methylpyrimidin-2-amine, 5-methyl3-arylpyrazolo[1,5-a]pyrimidines, and 5-methyl-2-R-pyrido[2,3-d]pyrimidin-4(3H)-ones containing a 5-amino-1,2,4-thiadiazole fragment linearly bound at position 3.

PAGES

1008-1012

Identifiers

URI

http://scigraph.springernature.com/pub.10.1007/s11172-016-1404-1

DOI

http://dx.doi.org/10.1007/s11172-016-1404-1

DIMENSIONS

https://app.dimensions.ai/details/publication/pub.1044640147


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