A convenient approach to the synthesis of 1-halomethyl-substituted 2,4,5,6-tetrahydro-1H-imidazo[1,2-a][1]benzazepines View Full Text


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Article Info

DATE

2021-12

AUTHORS

Ivanna Yu. Danyliuk, Valentyna S. Tolmachova, Eduard B. Rusanov, Mikhailo V. Vovk

ABSTRACT

Intramolecular halocyclization of N-allyl-4,5-dihydro-3H-1-benzazepin-2-amines, obtained by consecutive methylation and allylamination of benzazepin-2-ones, by the action of N-iodo(bromo)succinimide in acetonitrile at room temperature lead to the formation 1-(iodo(bromo)methyl)-2,4,5,6-tetrahydro-1H-imidazo[1,2-a][1]benzazepines in high yields.

PAGES

1187-1194

References to SciGraph publications

Identifiers

URI

http://scigraph.springernature.com/pub.10.1007/s10593-021-03042-x

DOI

http://dx.doi.org/10.1007/s10593-021-03042-x

DIMENSIONS

https://app.dimensions.ai/details/publication/pub.1145018227


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