Nucleophilic acylation of benzimidazole View Full Text


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Article Info

DATE

1983-01

AUTHORS

B. I. Khristich, A. M. Simonov, E. N. Shepelenko, V. A. Yatsimirskii

ABSTRACT

Conditions that make it possible to realize the direct C(2) acylation of benzimidazole and some of its derivatives were found. It is shown that bis products, which are converted to 2-acylbenzimidazoles upon heating to 140–200 °C with acyl halides in the presence of triethylamine, are formed in attempts to carry out C(2) acylation. More... »

PAGES

87-90

Identifiers

URI

http://scigraph.springernature.com/pub.10.1007/bf00512823

DOI

http://dx.doi.org/10.1007/bf00512823

DIMENSIONS

https://app.dimensions.ai/details/publication/pub.1053129752


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