Prodrug derivatives of (E)-N-methyl-N-((3-M ethylbenzofuran-2-yl)methyl)-3-(7-oxo-5,6,7,8-tetrahydro-1,8-naphthyridin-3-yl)acrylamide


Ontology type: sgo:Patent     


Patent Info

DATE

N/A

AUTHORS

John J. Partridge , John Colucci , Yves Gareau , Michel Therien , Robert Zamboni , Barry Hafkin , Anthony Marfat , Helmi Zaghdane

ABSTRACT

In part, the present disclosure is directed to prodrug derivatives of (E)-N-methyl-N-((3-methylbenzofuran-2-yl)methyl)-3-(7-oxo-5,6,7,8-tetrahydro-1,8-naphthyridin-3-yl)acrylamide compounds with significant solubility and bioavailability profiles.

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